BDBM412513 (Z)-N-(5-(1-(4-bromophenyl)prop-1- en-1-yl)pyrazin-2-yl)-5-fluoro-4- methylnicotinamide::US10399967, Compound 146

SMILES C\C=C(\c1ccc(Br)cc1)c1cnc(NC(=O)c2cncc(F)c2C)cn1

InChI Key InChIKey=LPNGUNKXNPYWTD-CQPUUCJISA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 412513   

TargetInterleukin-2(Homo sapiens (Human))
Prcl Research

US Patent
LigandPNGBDBM412513((Z)-N-(5-(1-(4-bromophenyl)prop-1- en-1-yl)pyrazin...)
Affinity DataIC50:  18nMAssay Description:Human peripheral blood mononuclear cells (PBMCs) are prepared from heparinized human blood by separation over a Ficoll density gradient.PBMCs are sti...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent