BDBM425068 3,4-dichloro-N-((S)-4-((1R,2S)-2-(4- fluorophenyl)-cyclopropylamino)-1-(4- (methylsulfonyl)piperazin-1-yl)-1- oxobutan-2-yl)benzamide::US10519118, Example 146::US10519118, Example 149::US11230534, Example 149
SMILES CS(=O)(=O)N1CCN(CC1)C(=O)[C@H](CCN[C@@H]1C[C@H]1c1ccc(F)cc1)NC(=O)c1ccc(Cl)c(Cl)c1
InChI Key InChIKey=RPXVSAGJFRPJAW-AJSBUHFISA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 425068
Affinity DataIC50: 7.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+4nMAssay Description:The KDM1A demethylase enzyme activity can obtained from mammalian cells or tissues expressing KDM1A from an endogenous or recombinant gene and purifi...More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:The KDM1A demethylase enzyme activity can obtained from mammalian cells or tissues expressing KDM1A from an endogenous or recombinant gene and purifi...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+4nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair