BDBM430282 US10556892, Compound 19::US10556892, Compound 8

SMILES CCS(=O)(=O)c1ccccc1C(=O)N1CCN(C[C@@H]1C)c1nc2ccc(F)cc2s1

InChI Key InChIKey=UKQOLPNYRVPCBM-AWEZNQCLSA-N

Data  6 IC50

PDB links: 2 PDB IDs match this monomer.

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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 430282   

TargetN-acylethanolamine-hydrolyzing acid amidase(Homo sapiens (Human))
The Regents of The University of California

US Patent
LigandPNGBDBM430282(US10556892, Compound 19 | US10556892, Compound 8)
Affinity DataIC50:  500nMAssay Description:HEK293 cells stably transfected with the human NAAA coding sequence cloned from a human spleen cDNA library (catalog no. 639124, Clontech, Mountain V...More data for this Ligand-Target Pair
TargetN-acylethanolamine-hydrolyzing acid amidase(Homo sapiens (Human))
The Regents of The University of California

US Patent
LigandPNGBDBM430282(US10556892, Compound 19 | US10556892, Compound 8)
Affinity DataIC50:  230nMAssay Description:HEK293 cells stably transfected with the human NAAA coding sequence cloned from a human spleen cDNA library (catalog no. 639124, Clontech, Mountain V...More data for this Ligand-Target Pair
TargetN-acylethanolamine-hydrolyzing acid amidase(Homo sapiens (Human))
The Regents of The University of California

US Patent
LigandPNGBDBM430282(US10556892, Compound 19 | US10556892, Compound 8)
Affinity DataIC50:  230nMAssay Description:Inhibition of human NAAAMore data for this Ligand-Target Pair
TargetN-acylethanolamine-hydrolyzing acid amidase(Homo sapiens (Human))
The Regents of The University of California

US Patent
LigandPNGBDBM430282(US10556892, Compound 19 | US10556892, Compound 8)
Affinity DataIC50:  228nMAssay Description:HEK293 cells stably transfected with the human NAAA coding sequence cloned from a human spleen cDNA library (catalog no. 639124, Clontech, Mountain V...More data for this Ligand-Target Pair
TargetN-acylethanolamine-hydrolyzing acid amidase(Homo sapiens (Human))
The Regents of The University of California

US Patent
LigandPNGBDBM430282(US10556892, Compound 19 | US10556892, Compound 8)
Affinity DataIC50:  230nMAssay Description:Inhibition of NAAA (unknown origin)More data for this Ligand-Target Pair
TargetN-acylethanolamine-hydrolyzing acid amidase(Homo sapiens (Human))
The Regents of The University of California

US Patent
LigandPNGBDBM430282(US10556892, Compound 19 | US10556892, Compound 8)
Affinity DataIC50:  554nMAssay Description:HEK293 cells stably transfected with the human NAAA coding sequence cloned from a human spleen cDNA library (catalog no. 639124, Clontech, Mountain V...More data for this Ligand-Target Pair