BDBM432087 US10577308, Compound 558
SMILES Cc1cccc(C)c1OCCCNCc1cccc(c1)-c1cncnc1
InChI Key InChIKey=UUJCWXBORMXXGI-UHFFFAOYSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 432087
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
The Florey Institute
US Patent
The Florey Institute
US Patent
Affinity DataIC50: 1.20E+3nMAssay Description:Test Protocol for Determining the Potency of Compounds on Nav1.2 and Nav1.6 Subtypes of Voltage-Gated Sodium Ion Channels Expressed in Mammalian Cell...More data for this Ligand-Target Pair
TargetSodium channel protein type 8 subunit alpha(Homo sapiens (Human))
The Florey Institute
US Patent
The Florey Institute
US Patent
Affinity DataIC50: 400nMAssay Description:Test Protocol for Determining the Potency of Compounds on Nav1.2 and Nav1.6 Subtypes of Voltage-Gated Sodium Ion Channels Expressed in Mammalian Cell...More data for this Ligand-Target Pair
TargetSodium channel protein type 8 subunit alpha(Homo sapiens (Human))
The Florey Institute
US Patent
The Florey Institute
US Patent
Affinity DataIC50: 300nMAssay Description:Test Protocol for Determining the Potency of Compounds on Nav1.2 and Nav1.6 Subtypes of Voltage-Gated Sodium Ion Channels Expressed in Mammalian Cell...More data for this Ligand-Target Pair
TargetSodium channel protein type 8 subunit alpha(Homo sapiens (Human))
The Florey Institute
US Patent
The Florey Institute
US Patent
Affinity DataIC50: 300nMAssay Description:Test Protocol for Determining the Potency of Compounds on Nav1.2 and Nav1.6 Subtypes of Voltage-Gated Sodium Ion Channels Expressed in Mammalian Cell...More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
The Florey Institute
US Patent
The Florey Institute
US Patent
Affinity DataIC50: 200nMAssay Description:Test Protocol for Determining the Potency of Compounds on Nav1.2 and Nav1.6 Subtypes of Voltage-Gated Sodium Ion Channels Expressed in Mammalian Cell...More data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
The Florey Institute
US Patent
The Florey Institute
US Patent
Affinity DataIC50: 200nMAssay Description:Test Protocol for Determining the Potency of Compounds on Nav1.2 and Nav1.6 Subtypes of Voltage-Gated Sodium Ion Channels Expressed in Mammalian Cell...More data for this Ligand-Target Pair