BDBM434142 US10562891, Example 64::US11008308, Example 65
SMILES Cc1cccc2c1nc(CS[C@@H]1CC[C@H](CN)CC1)[nH]c2=O
InChI Key
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 434142
TargetProtein mono-ADP-ribosyltransferase PARP14 [1611-1801](Homo sapiens (Human))
Ribon Therapeutics
US Patent
Ribon Therapeutics
US Patent
Affinity DataIC50: <1.00E+3nMAssay Description:Enzymatic inhibition of PARP14 was measured using a dissociation-enhanced lanthanide fluorescence immunoassay (DELFIA) monitoring the auto-modificati...More data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Enzymatic inhibition of PARP14 was measured using a dissociation-enhanced lanthanide fluorescence immunoassay (DELFIA) monitoring the auto-modificati...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Enzymatic inhibition of PARP14 was measured using a dissociation-enhanced lanthanide fluorescence immunoassay (DELFIA) monitoring the auto-modificati...More data for this Ligand-Target Pair