BDBM463500 2-(Benzo[d][1,3]dioxol-5-yl)-3-((S)-2-methylpyrrolidin-1-yl)quinoxaline-6-carboxylic acid::US10781185, Example 83::US11459307, Example 83
SMILES C[C@H]1CCCN1c1nc2cc(ccc2nc1-c1ccc2OCOc2c1)C(O)=O
InChI Key InChIKey=SEQCVAKNODWCHG-LBPRGKRZSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 463500
TargetPAS domain-containing serine/threonine-protein kinase(Homo sapiens (Human))
Bioenergenix
US Patent
Bioenergenix
US Patent
Affinity DataIC50: <1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
TargetPAS domain-containing serine/threonine-protein kinase(Homo sapiens (Human))
Bioenergenix
US Patent
Bioenergenix
US Patent
Affinity DataIC50: <1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
TargetPAS domain-containing serine/threonine-protein kinase [879-1323](Homo sapiens (Human))
Bioenergenix
US Patent
Bioenergenix
US Patent
Affinity DataIC50: <1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
TargetPAS domain-containing serine/threonine-protein kinase(Homo sapiens (Human))
Bioenergenix
US Patent
Bioenergenix
US Patent
Affinity DataIC50: <1.00E+3nMAssay Description:Compound screening was done via the following method. 10 mM stock solution of test compound in DMSO was prepared by dissolving test compound in DMSO ...More data for this Ligand-Target Pair