BDBM469032 US10807974, Example 43::US10995088, Example 43::US11608330, Example 43
SMILES NCc1ccc(s1)S(=O)(=O)c1cccc(c1)S(=O)(=O)N1CCC[C@H]1CO
InChI Key InChIKey=UOZFNARYACXBHE-LBPRGKRZSA-N
Data 9 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 469032
TargetProtein-lysine 6-oxidase(Sus scrofa)
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
Affinity DataIC50: 420nMAssay Description:LOX enzyme was obtained from pig skin by the method of Shackleton et al 1990.More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
Affinity DataIC50: >1.00E+5nMAssay Description:MAO-Glo Assay Kit: Promega, Cat No. V1402, MAO-A Enzyme: Promega, Cat No. V1452.More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
Affinity DataIC50: >1.00E+5nMAssay Description:MAO-Glo Assay Kit: Promega, Cat No. V1402, MAO-B Enzyme: Sigma, Cat No. M7441.More data for this Ligand-Target Pair
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
Affinity DataIC50: 420nMAssay Description:The following reagents were prepared:Reagents500 mM CHES, pH 9 (with NaOH), filtered (MW=207.29)20.7 g in 200 ml in dH2O10% Pluronic F-127 (store at ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
Affinity DataIC50: >1.00E+5nMAssay Description:Promega ROS-Glo H2O2 Assay Kit, 50 ml. Cat No. G8821Inhibitors (Test compounds):10 mM stock diluted to 10, 3, 1, 0.3, 0.1, 0.03, 0.01, 0.003, 0.001, ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
Affinity DataIC50: >1.00E+5nMAssay Description:The following reagents were prepared:ReagentsMAO-Glo Assay Kit: Promega, Cat No. V1402MAO-B Enzyme: Sigma, Cat No. M7441Deprenyl: Sigma, Cat No. M003...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Sus scrofa)
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
Affinity DataIC50: 420nMAssay Description:LOX enzyme was obtained from pig skin by the method of Shackleton et al 1990.Assay Plates:Black, flat bottom 96 well platesProcedure:1. Dilute LOX en...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
Affinity DataIC50: >1.00E+5nMAssay Description:MAO-B Enzyme: Sigma, Cat No. M7441Deprenyl: Sigma, Cat No. M003Assay Plates: 96 well white polystyrene, flat bottom plates, no lid: Fisher, Cat No. D...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
The Institute Of Cancer Research: Royal Cancer Hospital
US Patent
Affinity DataIC50: >1.00E+5nMAssay Description:The following reagents were prepared:ReagentsMAO-Glo Assay Kit: Promega, Cat No. V1402MAO-A Enzyme: Promega, Cat No. V1452Clorgyline: Sigma, Cat No. ...More data for this Ligand-Target Pair