BDBM469183 5-[2-cyclopropyl-5-(methylsulfonylmethyl)-1,3- benzoxazol-7-yl]-3-methoxy-1- methylpyridin-2-one::US10807982, Example 63
SMILES COc1cc(cn(C)c1=O)-c1cc(CS(C)(=O)=O)cc2nc(oc12)C1CC1
InChI Key InChIKey=IAQZFUGDAMBYAK-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469183
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair