BDBM470587 US10815244, Example T

SMILES COc1cc2ncnc(Nc3ccc(O[C@H]4CO[C@@H]5[C@@H](O)CO[C@H]45)c(Cl)c3)c2cc1OC

InChI Key InChIKey=LMWDCCYLPLDXQG-JWOSDPRPSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 470587   

TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM470587(US10815244, Example T)
Affinity DataIC50:  5.30nMAssay Description:In vitro inhibitory effect of histamine H3 antagonist on the electrically evoked contractile response of isolated guinea pig jejunum segments.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM470587(US10815244, Example T)
Affinity DataIC50: >100nMAssay Description:Briefly, the assay method measures ADP formed from EGFR kinase activity using luminescence derived from ATP-Luciferase detection system. Purified EGF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent