BDBM47103 US8937068, 124::US8937068, 193

SMILES CCNC(=O)Nc1ccc2ncc(nc2n1)-c1ccc(O)c(OC)c1

InChI Key InChIKey=OVGNDEJGXTVQKL-UHFFFAOYSA-N

Data  8 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 47103   

TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Zentaris

US Patent
LigandPNGBDBM47103(US8937068, 124 | US8937068, 193)
Affinity DataIC50:  212nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM47103(US8937068, 124 | US8937068, 193)
Affinity DataIC50:  2.20E+3nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Zentaris

US Patent
LigandPNGBDBM47103(US8937068, 124 | US8937068, 193)
Affinity DataIC50: >1.00E+5nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8/9(Homo sapiens (Human))
Zentaris

US Patent
LigandPNGBDBM47103(US8937068, 124 | US8937068, 193)
Affinity DataIC50:  1.00E+3nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Zentaris

US Patent
LigandPNGBDBM47103(US8937068, 124 | US8937068, 193)
Affinity DataIC50:  62nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM47103(US8937068, 124 | US8937068, 193)
Affinity DataIC50:  490nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Zentaris

US Patent
LigandPNGBDBM47103(US8937068, 124 | US8937068, 193)
Affinity DataIC50: >1.00E+5nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMitogen-activated protein kinase 8/9(Homo sapiens (Human))
Zentaris

US Patent
LigandPNGBDBM47103(US8937068, 124 | US8937068, 193)
Affinity DataIC50:  1.50E+3nMAssay Description:The inhibitory effect of the compounds according to the invention was tested on various serine/threonine, tyrosine and lipid kinases in enzymatic ass...More data for this Ligand-Target Pair
In DepthDetails US Patent