BDBM472877 Methyl 4-((4-(((2-(5-bromothiophen-2- yl))cyclopropyl)amino)methyl)- 4-fluoropiperidin-1-yl)methyl) benzoate::US10836743, Compound A103
SMILES COC(=O)c1ccc(CN2CCC(F)(CNC3CC3c3ccc(Br)s3)CC2)cc1
InChI Key InChIKey=JIVSPAJEIFWQIH-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 472877
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Shanghai Institute of Material Medica, Chinese Academy of Sciences
US Patent
Shanghai Institute of Material Medica, Chinese Academy of Sciences
US Patent
Affinity DataIC50: 80.5nMAssay Description:Screening method: lysine-specific demethylase 1 (LSD1) activity screeningInstrument: microplate reader Envision™ (PerkinElmer, USA).MATERIALS: Human ...More data for this Ligand-Target Pair