BDBM481786 3-((4-(4-chlorophenethyl)-5- oxo-4,5-dihydro-1,3,4- oxadiazol-2-yl)methyl)-5- methyl-4-oxo-3,4- dihydropyrido[2,3- d]pyrimidine-7-carbonitrile::US10913742, Example 28
SMILES Cc1cc(nc2ncn(Cc3nn(CCc4ccc(Cl)cc4)c(=O)o3)c(=O)c12)C#N
InChI Key InChIKey=PZLMINJQTMOPFT-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 481786
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 9nMAssay Description:The IC50 (effective concentration) of compounds on the human and rat TRPA1 channels were determined using a FLIPR Tetra instrument. CHO cells express...More data for this Ligand-Target Pair