BDBM481843 5-methyl-3-[[5-oxo-4-[rac- (2R)-2-(4-chlorophenyl)-2- fluoro-ethyl]-1,3,4-oxadiazol- 2-yl]methyl]pyrido[3,2- d]pyrimidine-4,6-dione::US10913742, Example 87
SMILES Cn1c2c(ccc1=O)ncn(Cc1nn(C[C@H](F)c3ccc(Cl)cc3)c(=O)o1)c2=O
InChI Key InChIKey=LFYAILSQQZVGPM-ZDUSSCGKSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 481843
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 43.8nMAssay Description:The IC50 (effective concentration) of compounds on the human and rat TRPA1 channels were determined using a FLIPR Tetra instrument. CHO cells express...More data for this Ligand-Target Pair