BDBM482299 US10919843, Compound VIII

SMILES CCCCCC1=C(NCc2ccccc2)C(=O)C([C@@H]2C=C(C)CC[C@H]2C(C)=C)=C(O)C1=O

InChI Key InChIKey=NTGIXJASMBWXRO-JTHBVZDNSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 482299   

TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Emerald Health Pharmaceuticals

US Patent
LigandPNGBDBM482299(US10919843, Compound VIII)
Affinity DataEC50:  1.40E+3nMAssay Description:HaCaT-EPO-Luc cells were maintained at 37° C. in a humidified atmosphere containing 5% CO2 in DMEM supplemented with 10% fetal calf serum (FBS), and ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
Emerald Health Pharmaceuticals

US Patent
LigandPNGBDBM482299(US10919843, Compound VIII)
Affinity DataEC50:  2.60E+3nMAssay Description:NIH3T3-EPO-luc cells were maintained at 37° C. in a humidified atmosphere containing 5% CO2 in DMEM supplemented with 10% fetal calf serum (FBS), and...More data for this Ligand-Target Pair
In DepthDetails US Patent