BDBM495071 US10995084, Ex. No. 3A-8
SMILES Cc1cccc(c1)[C@@H]1CC[C@@H](N1C(=O)CNC(=O)c1ccc(Cc2cc(C)n[nH]c2=O)c(C)c1)C(C)(C)C#N
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 495071
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Kissei Pharmaceutical
US Patent
Kissei Pharmaceutical
US Patent
Affinity DataKi: 0.0200nMAssay Description:The binding affinity assay of compounds for human CGRP receptor was carried out by inhibition of radiolabeled ligand [125I]-CGRP binding in human neu...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Kissei Pharmaceutical
US Patent
Kissei Pharmaceutical
US Patent
Affinity DataIC50: 0.360nMAssay Description:The binding affinity assay of compounds for human CGRP receptor was carried out by inhibition of radiolabeled ligand [125I]-CGRP binding in human neu...More data for this Ligand-Target Pair