BDBM50002805 (daltroban){4-[2-(4-Chloro-benzenesulfonylamino)-ethyl]-phenyl}-acetic acid::BM 13505::BM-13505::CHEMBL71685::Daltroban::{4-[2-(4-Chloro-benzenesulfonylamino)-ethyl]-phenyl}-acetic acid
SMILES OC(=O)Cc1ccc(CCNS(=O)(=O)c2ccc(Cl)cc2)cc1
InChI Key InChIKey=IULOBWFWYDMECP-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50002805
TargetThromboxane A2 receptor(Homo sapiens (Human))
Squibb Institute For Medical Research
Curated by PDSP Ki Database
Squibb Institute For Medical Research
Curated by PDSP Ki Database
TargetThromboxane A2 receptor(Homo sapiens (Human))
Squibb Institute For Medical Research
Curated by PDSP Ki Database
Squibb Institute For Medical Research
Curated by PDSP Ki Database
TargetThromboxane A2 receptor(Homo sapiens (Human))
Squibb Institute For Medical Research
Curated by PDSP Ki Database
Squibb Institute For Medical Research
Curated by PDSP Ki Database
Affinity DataKi: 63nMAssay Description:Compound was tested for its binding affinity at Thromboxane A2/ Prostaglandin H2 receptor by measuring its ability to displace [3H]-U-46,619 from gui...More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:In vitro thromboxane A2 antagonistic activity of the compound on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees centigradeMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
Squibb Institute For Medical Research
Curated by PDSP Ki Database
Squibb Institute For Medical Research
Curated by PDSP Ki Database
Affinity DataIC50: 460nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
Squibb Institute For Medical Research
Curated by PDSP Ki Database
Squibb Institute For Medical Research
Curated by PDSP Ki Database
Affinity DataIC50: 150nMAssay Description:In vitro thromboxane-A2 receptor binding affinity to displace by 50% [3H]-SQ 29548 binding from washed human plateletsMore data for this Ligand-Target Pair