BDBM50007594 CHEMBL3238295
SMILES COc1ccc(OC[C@](C)(O)C(=O)N2CCc3c2cccc3C#N)c(F)c1
InChI Key InChIKey=GZWMIPIQOGEGRP-FQEVSTJZSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50007594
Affinity DataEC50: 2.90nMAssay Description:Agonist activity at human AR expressed in CV1 cells after 17 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 427nMAssay Description:Displacement of [3H]mibolerone from full length human AR expressed in COS cells after 3.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity to human AR NTD (1 to 561 aa) expressed in CV1 cells coexpressing human AR-LBD (644-919 aa) assessed as N/C-termini interaction by a...More data for this Ligand-Target Pair