BDBM50017226 (R)-2-Amino-7-phosphono-heptanoic acid::2-Amino-7-phosphono-heptanoic acid::CHEMBL302783

SMILES N[C@H](CCCCCP(O)(O)=O)C(O)=O

InChI Key InChIKey=MYDMWESTDPJANS-ZCFIWIBFSA-N

Data  3 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50017226   

TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50017226((R)-2-Amino-7-phosphono-heptanoic acid | 2-Amino-7...)
Affinity DataKi:  490nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50017226((R)-2-Amino-7-phosphono-heptanoic acid | 2-Amino-7...)
Affinity DataKi:  4.14E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50017226((R)-2-Amino-7-phosphono-heptanoic acid | 2-Amino-7...)
Affinity DataKi:  6.42E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Homo sapiens (Human))TBA
LigandPNGBDBM50017226((R)-2-Amino-7-phosphono-heptanoic acid | 2-Amino-7...)
Affinity DataIC50:  850nMAssay Description:Inhibition of FTO (unknown origin) demethylation activity using m6A7-Broccoli RNA as substrate incubated for 3 mins under shaking condition and measu...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetRNA demethylase ALKBH5(Homo sapiens)TBA
LigandPNGBDBM50017226((R)-2-Amino-7-phosphono-heptanoic acid | 2-Amino-7...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of ALKBH5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed