BDBM50017479 2-(5,9-Diamino-2-methyl-4-oxo-nonanoylamino)-3-phenyl-propionic acid::CHEMBL28708

SMILES CC(CC(=O)[C@@H](N)CCCCN)C(=O)NC(Cc1ccccc1)C(O)=O

InChI Key InChIKey=NIMLXPSSVMNDFV-SIWZUTFBSA-N

Data  4 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50017479   

TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017479(2-(5,9-Diamino-2-methyl-4-oxo-nonanoylamino)-3-phe...)
Affinity DataKi:  2.00E+3nMAssay Description:Non-competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the intercept effect(Kii)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017479(2-(5,9-Diamino-2-methyl-4-oxo-nonanoylamino)-3-phe...)
Affinity DataKi:  2.80E+3nMAssay Description:Non-competitive inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the intercept effect(Kii)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase B(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017479(2-(5,9-Diamino-2-methyl-4-oxo-nonanoylamino)-3-phe...)
Affinity DataKi:  8.80E+3nMAssay Description:Competitive inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017479(2-(5,9-Diamino-2-methyl-4-oxo-nonanoylamino)-3-phe...)
Affinity DataKi:  2.10E+5nMAssay Description:Inhibition of aminopeptidase M or membrane leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017479(2-(5,9-Diamino-2-methyl-4-oxo-nonanoylamino)-3-phe...)
Affinity DataIC50: >5.00E+5nMAssay Description:Competitive inhibition of leucine aminopeptidase; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed