BDBM50019122 CHEMBL3288417

SMILES COc1ccc2n(c(CCn3c4ncccc4n(C)c3=O)nc2c1)-c1ccccn1

InChI Key InChIKey=PMUJUEIYPOAHHW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50019122   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Homo sapiens (Human))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50019122(CHEMBL3288417)
Affinity DataIC50:  220nMAssay Description:Inhibition of human recombinant PDE10A expressed in Sf9 insect cell system assessed as inhibition of cAMP hydrolysis preincubated for 30 mins before ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed