BDBM50019130 CHEMBL3288425

SMILES COc1ccc2[nH]c(CCc3nc(C)c4ccccn34)nc2c1

InChI Key InChIKey=VJERNBDIQMOLMN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50019130   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Homo sapiens (Human))
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50019130(CHEMBL3288425)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human recombinant PDE10A expressed in Sf9 insect cell system assessed as inhibition of cAMP hydrolysis preincubated for 30 mins before ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed