BDBM50025030 CHEMBL3355097
SMILES [Br-].[Br-].[H][C@]12N3\C=C4/[C@]5([H])N(\C=C1\[C@@]1([H])C[C@@]6([H])[C@@]2(CC[N+]6(Cc2ccc(cc2)[N+]([O-])=O)C[C@H]1CC)c1ccccc31)c1ccccc1[C@@]51CC[N+]2(Cc3ccc(cc3)[N+]([O-])=O)C[C@@H](CCO)[C@]4([H])C[C@@]12[H]
InChI Key InChIKey=CSHQOJIGRNCSBW-IMPULFQBSA-L
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50025030
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 32nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 4.17E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataEC50: 32nMAssay Description:Displacement of [3H]NMS from pig muscarinic M2 receptor after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in GH3 cells by Ca2+/Fluo-4 assayMore data for this Ligand-Target Pair