BDBM50027177 Cilostamide

SMILES CN(C1CCCCC1)C(=O)CCCOc1ccc2nc(O)ccc2c1

InChI Key InChIKey=UIAYVIIHMORPSJ-UHFFFAOYSA-N

Data  3 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50027177   

LigandPNGBDBM50027177(Cilostamide)
Affinity DataIC50: 170nMAssay Description:In vitro inhibition of cyclic AMP phosphodiesterase from human platelets.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
The Baruch S. Blumberg Institute

Curated by ChEMBL
LigandPNGBDBM50027177(Cilostamide)
Affinity DataIC50: 27nMAssay Description:Inhibition of human recombinant PDE3 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50027177(Cilostamide)
Affinity DataKi:  5nMAssay Description:Binding affinity for low Km cAMP phosphodiesterase PDE III of human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50027177(Cilostamide)
Affinity DataKi:  20nMAssay Description:Inhibition of human phosphodiesterase 3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50027177(Cilostamide)
Affinity DataKi:  2.20E+4nMAssay Description:Binding affinity for [Ca(2+)]/calmodulin dependent phosphodiesterase PDE 1 of human brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed