BDBM50029188 CHEMBL2165920
SMILES CC(C)C[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](N)C(C)C)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc1ccccc1)C(N)=O
InChI Key InChIKey=JFZCLMZUABKABL-GVCDGELBSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50029188
Affinity DataKi: 0.0100nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Displacement of [125I]YVP from human NPFFR1 expressed in CHO cells by gamma-counter methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF2 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [125I]YVP from human NPFFR1 expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [125I]EYF from human NPFFR2 expressed in CHO cells by gamma-counter methodMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Agonist activity at human NPFF1R expressed in HEK293 cells by dynamic mass redistribution assayMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at human NPFF1 receptor expressed in HEK293 cells assessed as reduction in forskolin- stimulated cAMP levelMore data for this Ligand-Target Pair