BDBM50067251 4-{(E)-2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-8-yloxymethyl)-2,4-dichloro-phenyl]-methyl-carbamoyl}-methyl)-carbamoyl]-vinyl}-N,N-dimethyl-benzamide; hydrochloride::CHEMBL543899
SMILES CN(C)C(=O)c1ccc(\C=C\C(=O)NCC(=O)N(C)c2ccc(Cl)c(COc3cccn4c(Br)c(C)nc34)c2Cl)cc1
InChI Key InChIKey=NDOBHDUXUJNXHX-NTEUORMPSA-N
Data 5 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50067251
Affinity DataIC50: 0.660nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Concentration required to inhibit specific binding of [3H]BK (1.2 nM) to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B2...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition specific binding of [3H]BK (1.0 nM) to human Bradykinin receptor B2 which was expressed in CHO (Chinese hamster ovary) cells by 50%.More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B...More data for this Ligand-Target Pair
Affinity DataIC50: 0.660nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair