BDBM50072448 CHEMBL18767::{(3-Carbamimidoyl-phenyl)-[3-(2'-sulfamoyl-biphenyl-4-yl)-propyl]-amino}-acetic acid methyl ester; TFA
SMILES COC(=O)CN(CCCc1ccc(cc1)-c1ccccc1S(N)(=O)=O)c1cccc(c1)C(N)=N
InChI Key InChIKey=WTZPFQZXGTVVPM-UHFFFAOYSA-N
Data 7 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50072448
Affinity DataKi: 1.30nMAssay Description:Inhibition of serine protease factor Xa enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity against Coagulation factor X in an enzyme inhibition assay.More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Inhibition of serine protease trypsin enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition of serine protease thrombin enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Compound was tested for the inhibition of serine protease plasmin enzyme.More data for this Ligand-Target Pair
Affinity DataKi: 4.20E+3nMAssay Description:Compound was tested for the inhibition of serine protease factor VIIa enzyme.More data for this Ligand-Target Pair
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by ChEMBL
Dupont Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 3.30E+4nMAssay Description:Compound was tested for the inhibition of serine protease tissue plasminogen activator enzyme.More data for this Ligand-Target Pair