BDBM50080387 (R)-1-{2-[1-(1-Methyl-1H-pyrrol-2-yl)-1-phenyl-meth-(E)-ylideneaminooxy]-ethyl}-piperidine-3-carboxylic acid; hydrochloride::CHEMBL553582
SMILES Cn1cccc1\C(=N\OCCN1CCC[C@H](C1)C(O)=O)c1ccccc1
InChI Key InChIKey=DATKEIYRWPELMK-RWNPKEDZSA-N
Data 1 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50080387
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair