BDBM50089398 CHEMBL3577981
SMILES [H][C@@]12CCCN1C(=O)[C@@]1([H])CCCN1C(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCNC(N)=N)NC2=O
InChI Key InChIKey=MTKQTEXYJKPBQD-GNDHHEKASA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 13 hits for monomerid = 50089398
Affinity DataKi: 20nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Displacement of MTII from mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse MC4R by alphascreen cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of [125I]-NDP-MSH from mouse melanocortin receptor 4 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...More data for this Ligand-Target Pair
Affinity DataIC50: 1.23E+4nMAssay Description:Displacement of [125I]-NDP-MSH from mouse melanocortin receptor 5 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of [125I]-NDP-MSH from human melanocortin receptor 4 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:Displacement of [125I]-NDP-MSH from mouse melanocortin receptor 3 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse MC3R by alphascreen cAMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.50E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by cAMP functional bioassayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+8nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by cAMP functional bioassayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Displacement of [125I]-NDP-MSH from mouse melanocortin receptor 1 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...More data for this Ligand-Target Pair