BDBM50096422 CHEMBL3577137

SMILES CCCCCCCC\C=C/CCCCCCCC(=O)OCCCOP(O)(=O)OC[C@H](N)C(O)=O

InChI Key InChIKey=MNVYCWBZLPRJPH-DYYZXQNHSA-N

Data  9 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50096422   

TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50:  25nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 34(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at GPR34 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50:  25nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 34(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50: >3.16E+3nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of ectodomain she...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50:  19nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 34(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50:  540nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 34(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50:  537nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 34(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096422(CHEMBL3577137)
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed