BDBM50117652 CHEMBL3613636

SMILES CCN(CC)C1CCN(CC1)S(=O)(=O)c1ccc(NC(=O)c2ccc(cc2)C(F)(F)F)cc1

InChI Key InChIKey=ZMZNMRJHXUNOEL-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50117652   

TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Renovis

Curated by ChEMBL

LigandBDBM50117652(CHEMBL3613636)Copy SMILESCopy InChI

Affinity DataIC50:  910nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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