BDBM50131688 (E)-4-(3,5-dimethoxystyryl)phenol::3,5-Dimethoxy-4'-hydroxyl-trans-stilbene::4'-hydroxy-3,5-dimethoxy stilbene::4-(3,5-dimethoxystyryl)phenol::4-[(E)-2-(3,5-Dimethoxy-phenyl)-vinyl]-phenol::4-[2-(3,5-Dimethoxy-phenyl)-vinyl]-phenol::CHEMBL83527::E 4-[2-(3,5-Dimethoxy-phenyl)-vinyl]-phenol::Pterostilben::Pterostilbene

SMILES COc1cc(OC)cc(\C=C\c2ccc(O)cc2)c1

InChI Key InChIKey=VLEUZFDZJKSGMX-ONEGZZNKSA-N

Data  2 KI  14 IC50  1 EC50

PDB links: 5 PDB IDs match this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50131688   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50131688((E)-4-(3,5-dimethoxystyryl)phenol | 3,5-Dimethoxy-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase of intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50131688((E)-4-(3,5-dimethoxystyryl)phenol | 3,5-Dimethoxy-...)
Affinity DataIC50:  7.50E+3nMAssay Description:Antagonist activity at rat TRPA1 expressed in HEK293 cells assessed as inhibition of allyl isothiocyanate-induced increase of intracellular calcium l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50131688((E)-4-(3,5-dimethoxystyryl)phenol | 3,5-Dimethoxy-...)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as induction of intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed