BDBM50143782 3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiophene-2-carboxylic acid (2,6-dimethyl-4-oxazol-2-yl-phenyl)-amide::CHEMBL59288

SMILES Cc1noc(NS(=O)(=O)c2ccsc2C(=O)Nc2c(C)cc(cc2C)-c2ncco2)c1Cl

InChI Key InChIKey=VDNHFRIBVSEFJN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50143782   

TargetEndothelin-1 receptor(RAT)
Encysive Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50143782(3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...)
Affinity DataIC50:  1.27nMAssay Description:Inhibitory concentration towards endothelin A receptor in rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed