BDBM50163091 6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1-(2-pyrrolidin-1-yl-ethyl)-1H-indol-5-yl]-amide::CHEMBL367088

SMILES Clc1nc2sccn2c1S(=O)(=O)Nc1ccc2n(CCN3CCCC3)ccc2c1

InChI Key InChIKey=QOOWDQCUBAWIJN-UHFFFAOYSA-N

Data  2 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50163091   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50163091(6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1...)
Affinity DataKi:  9.80nMAssay Description:Antagonist activity at human recombinant 5HT6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50163091(6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1...)
Affinity DataKi:  9.80nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50163091(6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1...)
Affinity DataIC50:  135nMAssay Description:Inhibition of human recombinant 5HT6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed