BDBM50167276 CHEMBL3798844
SMILES Fc1cc2n(-c3cccnc3)c3cn[nH]c3c2cc1F
InChI Key InChIKey=PEWYGTLRHLRPDV-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50167276
Affinity DataIC50: 50nMAssay Description:Inhibition of human CYP1A2 expressed in Escherichia coli DH5alphaMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:Inhibition of recombinant full-length human MetAP2 catalytic domain (110 to 478 residues) expressed in baculovirus using Met-AMC as substrate by fluo...More data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Inhibition of human MetAP2 in HUVEC cells assessed as accumulation of N-Met 14-3-3gamma after 24 hrs by western blot analysisMore data for this Ligand-Target Pair