BDBM50177071 3-(4-Ethyl-phenyl)-9-(2,2,2-trifluoro-ethylamino)-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one::9-(2',2',2'-Trifluoroethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one::CHEMBL376372
SMILES CCc1ccc(cc1)-n1cnc2c(sc3nccc(NCC(F)(F)F)c23)c1=O
InChI Key InChIKey=HVNDCFLLFFZJIK-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50177071
Affinity DataIC50: 99nMAssay Description:Antagonist activity at human mGluR1 expressed in 1321N1 cells assessed as effect on L-glutamate-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 99nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human mGluR5 expressed in 1321N1 cells assessed as effect on L-glutamate-induced calcium mobilizationMore data for this Ligand-Target Pair