BDBM50177074 9-(Ethyl-methyl-amino)-3-(4-ethyl-phenyl)-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one::9-(N,N-ethylmethylamino)-3-(4'-ethylphenyl)-3H-5-thia-1,3,6-triazafluoren-4-one::CHEMBL223543
SMILES CCN(C)c1ccnc2sc3c(ncn(-c4ccc(CC)cc4)c3=O)c12
InChI Key InChIKey=IPMMMSQQYJZTAG-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50177074
Affinity DataIC50: 37nMAssay Description:Antagonist activity at human mGluR1 expressed in 1321N1 cells assessed as effect on L-glutamate-induced calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
Affinity DataIC50: 2.57E+3nMAssay Description:Antagonist activity at human mGluR5 expressed in 1321N1 cells assessed as effect on L-glutamate-induced calcium mobilizationMore data for this Ligand-Target Pair