BDBM50177563 CHEMBL380855::N-((R)-3-(4-chlorophenyl)-1-(4-(2-(diethylamino)-1-(2-fluorophenyl)ethyl)piperazin-1-yl)-1-oxopropan-2-yl)-2-(isoindolin-1-yl)acetamide
SMILES CCN(CC)CC(N1CCN(CC1)C(=O)[C@@H](Cc1ccc(Cl)cc1)NC(=O)CC1NCc2ccccc12)c1ccccc1F
InChI Key InChIKey=AITZMTQUXXOZQF-QYEGGPJFSA-N
Data 4 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50177563
Affinity DataKi: 7.30nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC5R expressed in HEK293 cellMore data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC3R expressed in HEK293 cellMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from cloned human MC1R expressed in HEK293 cellMore data for this Ligand-Target Pair