BDBM50208926 CHEMBL3884179

SMILES C[C@H](N1C(=O)C(C)(C)c2cnc(Nc3cccnc3)nc12)c1ccc(F)cc1

InChI Key InChIKey=KWJOTUQSCIOUKF-ZDUSSCGKSA-N

Data  3 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50208926   

TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50208926(CHEMBL3884179)
Affinity DataIC50:  62nMAssay Description:Inhibition of full length human MARK3 using biotin labeled peptide substrate by HTRF based assayMore data for this Ligand-Target Pair
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50208926(CHEMBL3884179)
Affinity DataIC50:  61nMAssay Description:Inhibition of MARK3 (unknown origin)More data for this Ligand-Target Pair
TargetMAP/microtubule affinity-regulating kinase 4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50208926(CHEMBL3884179)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human MARK4 expressed in HEK293T cells coexpressing tau protein assessed as reduction in tau phosphorylation at Ser262 residues by Alph...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed