BDBM50209237 6-bromo-1H-indazole::CHEMBL247365
SMILES Brc1ccc2cn[nH]c2c1
InChI Key InChIKey=WMKDUJVLNZANRN-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50209237
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of rat neuronal NOSMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Eberhard Karls Universit£T T£Bingen
Curated by ChEMBL
Eberhard Karls Universit£T T£Bingen
Curated by ChEMBL
Affinity DataKd: 3.80E+4nMAssay Description:Binding affinity to human DYRK1A (127 to 485 residues) expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant by isothermal...More data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of NOS1More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Reversal inhibition of full length recombinant human MetAP2 expressed in baculovirus infected insect Sf9 cells using Met-AMC as substrate measured fo...More data for this Ligand-Target Pair