BDBM50216491 5-benzyl-6-(4-phenylpiperidin-1-yl)pyrimidine-2,4(1H,3H)-dione::CHEMBL230675
SMILES O=c1[nH]c(N2CCC(CC2)c2ccccc2)c(Cc2ccccc2)c(=O)[nH]1
InChI Key InChIKey=QKBURCBWLIXXPH-UHFFFAOYSA-N
Data 5 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50216491
Affinity DataKi: 8nMAssay Description:Displacement of [3H]dexamethasone from human recombinant glucocorticoid receptor expressed in baculovirus after 18 hrs by scintillation counting anal...More data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Displacement of [3H]dexamethasone from human recombinant GRMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Antagonist activity at human GRMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Antagonist activity at glucocorticoid receptor in human SW1353 cells assessed as inhibition of dexamethasone-induced luciferase expression after 16 h...More data for this Ligand-Target Pair
Affinity DataKi: 930nMAssay Description:Displacement of [3H]aldosterone from mineralocorticoid receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair