BDBM50232129 1-[5-(Cyano-isopropyl)-indan-1-yl]-3-(1H-indazol-4-yl)-urea::CHEMBL428061

SMILES CC(C)(C#N)c1cccc2C(CCc12)NC(=O)Nc1cccc2[nH]ncc12

InChI Key InChIKey=XOZDBVYABUEFNZ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50232129   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50232129(1-[5-(Cyano-isopropyl)-indan-1-yl]-3-(1H-indazol-4...)
Affinity DataIC50:  19nMAssay Description:Blockade of human TRPV1 receptor assessed as inhibition of capsaicin-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed