BDBM50232884 CHEMBL4060962
SMILES [H][C@]12C[C@@]3([H])C4=CCO[C@@]5([H])CC(=O)N6c7ccc(N)cc7[C@@]1(CCN2C4)[C@]6([H])[C@@]35[H]
InChI Key InChIKey=NRGHCWQGTHPFTE-FVWCLLPLSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50232884
Affinity DataKi: 18nMAssay Description:Displacement of [3H]strychnine from glycine receptor alpha 1 in rat brain synaptic membranesMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 275nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University In Cairo
Curated by ChEMBL
The German University In Cairo
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair