BDBM50238201 CHEMBL4065936
SMILES CCc1cc(ccc1\C=C1/SC(=O)NC1=O)-c1ccc(cc1OC)-n1c(C)cc(\C=C2/SC(=O)NC2=O)c1C
InChI Key InChIKey=KTUVABRLAOWXTO-CPGLPWGESA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50238201
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 177nMAssay Description:Inhibition of [3H][D-Ala2,D-Leu5]enkephalin binding to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
TargetGlutaminase liver isoform, mitochondrial(Homo sapiens)
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of recombinant human His-tagged GAB (P56 to V602 residues) expressed in Escherichia coli C41(DE3)pLysS using glutamine as substrate preinc...More data for this Ligand-Target Pair
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Inhibition of recombinant human His-tagged KGA (L123 to L669 residues) expressed in Escherichia coli BL21(DE3)pLysS using glutamine substrate preincu...More data for this Ligand-Target Pair