BDBM50239049 CHEMBL4086782
SMILES CCS(=O)(=O)c1ccc(Oc2cc3cc([nH]c3cc2C2CCC(=O)N2C)-c2ccc(cn2)C(F)(F)F)cc1
InChI Key InChIKey=NJMQGAPDEDUCFJ-UHFFFAOYSA-N
Data 4 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50239049
Affinity DataEC50: 1.70nMAssay Description:Activation of glucokinase in rat INS-1 cells assessed as increase in D-2-deoxyglucose-6-phosphate level in presence of D-2-deoxyglucose by HILIC LC-M...More data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Activation of recombinant human glucokinase assessed as conversion of D-glucose to D-glucose-6-phosphate in presence of 2.5 mM glucose by G6PDH coupl...More data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Inhibition of cAMP PDE II enzymeMore data for this Ligand-Target Pair
Affinity DataEC50: 174nMAssay Description:Inhibition of cGMP PDE II enzymeMore data for this Ligand-Target Pair