BDBM50240415 CHEMBL4078433
SMILES COc1ccc(cc1)S(=O)(=O)N(CC(=O)NO)Cc1cccc(c1)C(O)=O
InChI Key InChIKey=YBQPTPBTTDQLMD-UHFFFAOYSA-N
Data 9 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 50240415
Target72 kDa type IV collagenase(Homo sapiens (Human))
Fraunhofer Institute For Cell Therapy and Immunology Izi
Curated by ChEMBL
Fraunhofer Institute For Cell Therapy and Immunology Izi
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of APMA-activated recombinant human MMP2 expressed in CHO cells using Mca-PLGL-(DapDnp)-AR-NH2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Fraunhofer Institute For Cell Therapy and Immunology Izi
Curated by ChEMBL
Fraunhofer Institute For Cell Therapy and Immunology Izi
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of APMA-activated recombinant human MMP9 expressed in CHO cells using Mca-PLGL-(DapDnp)-AR-NH2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 10(Homo sapiens (Human))
Fraunhofer Institute For Cell Therapy and Immunology Izi
Curated by ChEMBL
Fraunhofer Institute For Cell Therapy and Immunology Izi
Curated by ChEMBL
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged ADAM10 expressed in baculovirus infected Sf21 cells using Abz-LANAVRSSSR-(DapDnp)-NH2 as subs...More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Fraunhofer Institute For Cell Therapy and Immunology Izi
Curated by ChEMBL
Fraunhofer Institute For Cell Therapy and Immunology Izi
Curated by ChEMBL
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of recombinant human C-terminal His6-tagged ADAM17 expressed in baculovirus infected Sf21 cells using Abz-LANAVRSSSR-(DapDnp)-NH2 as subst...More data for this Ligand-Target Pair
TargetMeprin A subunit beta(Homo sapiens)
Fraunhofer Institute For Cell Therapy And Immunology Izi
Curated by ChEMBL
Fraunhofer Institute For Cell Therapy And Immunology Izi
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of recombinant human meprin beta expressed in yeast using Abz-YVAEAPK(Dnp)G-OH as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetCollagenase 3(Homo sapiens (Human))
Fraunhofer Institute For Cell Therapy and Immunology Izi
Curated by ChEMBL
Fraunhofer Institute For Cell Therapy and Immunology Izi
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of APMA-activated recombinant human MMP13 expressed in mouse NS0 cells using Mca-PLGL-(DapDnp)-AR-NH2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetMeprin A subunit beta(Homo sapiens)
Fraunhofer Institute For Cell Therapy And Immunology Izi
Curated by ChEMBL
Fraunhofer Institute For Cell Therapy And Immunology Izi
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant human meprin beta expressed in yeast using Abz-YVAEAPK(Dnp)G-OH as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetMeprin A subunit alpha(Homo sapiens)
Fraunhofer Institute For Cell Therapy And Immunology Izi
Curated by ChEMBL
Fraunhofer Institute For Cell Therapy And Immunology Izi
Curated by ChEMBL
Affinity DataIC50: 3.29E+3nMAssay Description:Inhibition of recombinant human meprin alpha expressed in insect cells using Abz-YVADAPK(Dnp)G-OH as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetMeprin A subunit alpha(Homo sapiens)
Fraunhofer Institute For Cell Therapy And Immunology Izi
Curated by ChEMBL
Fraunhofer Institute For Cell Therapy And Immunology Izi
Curated by ChEMBL
Affinity DataIC50: 3.29E+3nMAssay Description:Inhibition of recombinant human meprin alpha expressed in S2 insect cells using Abz-YVADAPK(Dnp)G-OH as substrate by fluorescence assayMore data for this Ligand-Target Pair