BDBM50255292 CHEMBL4061423

SMILES N[C@@H](CCP(O)(=O)C(O)c1csc(c1)[N+]([O-])=O)C(O)=O

InChI Key InChIKey=GDELUTDICYGXSV-AADKRJSRSA-N

Data  8 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50255292   

TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50255292(CHEMBL4061423)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at mGlu6 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 7(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50255292(CHEMBL4061423)
Affinity DataEC50:  4.18E+5nMAssay Description:Agonist activity at mGlu7 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 8(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50255292(CHEMBL4061423)
Affinity DataEC50:  380nMAssay Description:Agonist activity at mGlu8 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as increase in intracellular calcium...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 8(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50255292(CHEMBL4061423)
Affinity DataEC50:  510nMAssay Description:Agonist activity at mGlu6 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as increase in intracellular calcium...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50255292(CHEMBL4061423)
Affinity DataEC50:  320nMAssay Description:Agonist activity at mGlu4 in Wistar rat striatum assessed as decrease in striatal GABAergic inhibitory post-synaptic potential by whole cell patch cl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50255292(CHEMBL4061423)
Affinity DataEC50:  9.32E+3nMAssay Description:Agonist activity at mGlu4 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50255292(CHEMBL4061423)
Affinity DataEC50:  190nMAssay Description:Agonist activity at mGlu4 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
University of Paris

Curated by ChEMBL
LigandPNGBDBM50255292(CHEMBL4061423)
Affinity DataEC50:  160nMAssay Description:Agonist activity at mGlu4 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed