BDBM50256075 2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-yl)-1-(piperidin-1-yl)ethanone::CHEMBL481886

SMILES Clc1ccc(-c2nn(CC(=O)N3CCCCC3)nc2-c2ccc(Cl)cc2Cl)c(Cl)c1

InChI Key InChIKey=XTLDZHVEQHHQBL-UHFFFAOYSA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50256075   

TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256075(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50:  169nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256075(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataIC50:  5.90nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Central University

Curated by ChEMBL
LigandPNGBDBM50256075(2-(4,5-bis(2,4-dichlorophenyl)-2H-1,2,3-triazol-2-...)
Affinity DataEC50:  122nMAssay Description:Antagonist activity at human CB1 receptor expressed in HEK293 cells assessed as inhibition of Eu-GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed