BDBM50260048 CHEMBL4084933
SMILES [Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[O-]S(=O)(=O)Oc1cc(OCc2ccc(COc3cc(OS([O-])(=O)=O)cc4oc(-c5ccc(OS([O-])(=O)=O)c(OS([O-])(=O)=O)c5)c(OS([O-])(=O)=O)c(=O)c34)cc2)c2c(c1)oc(-c1ccc(OS([O-])(=O)=O)c(OS([O-])(=O)=O)c1)c(OS([O-])(=O)=O)c2=O
InChI Key InChIKey=DDUSVFYSJIYYFC-UHFFFAOYSA-F
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 19 hits for monomerid = 50260048
Affinity DataIC50: 5.05E+5nMAssay Description:Inhibition of human F10a by using chromogenic substrate spectrozyme F10a preincubated for 5 mins followed by substrate addition by spectrophotometric...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30E+3nMAssay Description:Direct inhibition of human Lys-plasmin preincubated for 5 mins followed by Spectrozyme PL addition by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+6nMAssay Description:Inhibition of human F9a by using chromogenic substrate spectrozyme F9a preincubated for 5 mins followed by substrate addition by spectrophotometric m...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human F12a by using chromogenic substrate spectrozyme F12a preincubated for 5 mins followed by substrate addition by spectrophotometric...More data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMAssay Description:Allosteric inhibition of human plasmin using chromogenic substrate spectrozyme PL preincubated for 5 mins followed by substrate addition measured ove...More data for this Ligand-Target Pair
Affinity DataIC50: 1.56E+5nMAssay Description:Inhibition of human thrombin by using chromogenic substrate spectrozyme TH preincubated for 5 mins followed by substrate addition by spectrophotometr...More data for this Ligand-Target Pair
Affinity DataIC50: 2.59E+4nMAssay Description:Binding affinity to human plasmin assessed as loss of intrinsic tryptophan fluorescence at 250 uM by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+3nMAssay Description:Binding affinity to human dansyl-EGR-chloromethylketone-plasmin complex assessed as loss of intrinsic tryptophan fluorescence by spectrofluorometric ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+4nMAssay Description:Allosteric inhibition of full length human plasmin by using chromogenic substrate spectrozyme PL preincubated for 5 mins followed by substrate additi...More data for this Ligand-Target Pair
Affinity DataIC50: 8.80E+3nMAssay Description:Allosteric inhibition of human plasmin using chromogenic substrate spectrozyme PL preincubated for 5 mins followed by substrate addition measured ove...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30E+3nMAssay Description:Allosteric inhibition of human plasmin using chromogenic substrate spectrozyme PL preincubated for 5 mins followed by substrate addition measured ove...More data for this Ligand-Target Pair
Affinity DataKd: 4.40E+3nMAssay Description:Allosteric inhibition of human plasmin using chromogenic substrate spectrozyme PL preincubated for 5 mins followed by substrate addition measured ove...More data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+4nMAssay Description:Allosteric inhibition of human plasmin using chromogenic substrate spectrozyme PL preincubated for 5 mins followed by substrate addition measured ove...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Binding affinity to human plasmin assessed as loss of intrinsic tryptophan fluorescence at 250 uM by spectrofluorometric methodMore data for this Ligand-Target Pair
Affinity DataKd: 700nMAssay Description:Allosteric inhibition of full length human plasmin by using chromogenic substrate spectrozyme PL preincubated for 5 mins followed by substrate additi...More data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Allosteric inhibition of human plasmin assessed as delay in clot lysis after 410 mins by spectrophotometer methodMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of human neutrophil elastase using S1384 as substrate preincubated for 5 mins followed by substrate additionMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of human plasmin assessed as reduction in plasmin-mediated thrombin/factor 13a-induced clot fibrinolysis measured over 50 to 200 min by UV...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+5nMAssay Description:Inhibition of human F11a by using chromogenic substrate S-2366 preincubated for 5 mins followed by substrate addition by spectrophotometric methodMore data for this Ligand-Target Pair