BDBM50295287 2-(1-methyl-5-(4-methylbenzoyl)-1H-pyrrol-2-yl)acetic acid::CHEMBL1020::MCN-2559::TOLMETIN::Tolectin::[1-Methyl-5-(4-methyl-benzoyl)-1H-pyrrol-2-yl]-acetic acid::[1-Methyl-5-(4-methyl-benzoyl)-1H-pyrrol-2-yl]-acetic acid(tolmetin)

SMILES Cc1ccc(cc1)C(=O)c1ccc(CC(O)=O)n1C

InChI Key InChIKey=UPSPUYADGBWSHF-UHFFFAOYSA-N

Data  9 KI  2 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50295287   

TargetInterleukin-8(Homo sapiens (Human))
Grupo Uriach

Curated by ChEMBL
LigandPNGBDBM50295287(2-(1-methyl-5-(4-methylbenzoyl)-1H-pyrrol-2-yl)ace...)
Affinity DataIC50:  90nMAssay Description:Inhibition of CXCL8-induced chemotaxis in human polymorphonuclear leukocyte pretreated for 15 mins measured after 4 hrs by cell migration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed