BDBM50309995 4-((1H-1,2,4-Triazol-1-yl)methyl)-5-(4-bromophenyl)-N-(1-(4-bromophenyl)ethyl)-1-(2,4-dichlorophenyl)-1H-pyrazole-3-carboxamide::CHEMBL598549

SMILES Cc1cc(Br)ccc1CNC(=O)c1nn(c(c1Cn1cncn1)-c1ccc(Br)cc1)-c1ccc(Cl)cc1Cl

InChI Key InChIKey=MFICBBWNFIHARA-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50309995   

TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50309995(4-((1H-1,2,4-Triazol-1-yl)methyl)-5-(4-bromophenyl...)
Affinity DataIC50:  1.40nMAssay Description:Displacement of [3H]CP55,940 from CB1 receptor in Sprague-Dawley rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50309995(4-((1H-1,2,4-Triazol-1-yl)methyl)-5-(4-bromophenyl...)
Affinity DataIC50:  28.2nMAssay Description:Inverse agonist activity at human recombinant CB1 receptor expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50309995(4-((1H-1,2,4-Triazol-1-yl)methyl)-5-(4-bromophenyl...)
Affinity DataIC50:  6.48E+3nMAssay Description:Displacement of [3H]WIN55,212-2 from human recombinant CB2 receptor expressed in CHO-K1 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed